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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T13510 | Sigma-LIGAND-1 | Sigma receptor | |
Sigma-LIGAND-1 is a selective Sigma Receptor ligand with an IC50s of 16 nM, 19 nM at the DTG site and the PPP site, respectively. Sigma-LIGAND-1 has a Ki of 4000 nM at the dopamine D2 receptor. | |||
T63048 | Sigma-LIGAND-1 hydrochloride | ||
Sigma-LIGAND-1 hydrochloride is a selective sigma receptor ligand that acts at the DTG (IC50: 16 nM) and PPP (IC50: 19 nM) sites. Sigma-LIGAND-1 hydrochloride is able to act on the dopamine D2 receptor (Ki: 4000 nM). | |||
T39211 | PD 144418 oxalate | Sigma receptor | |
PD 144418 oxalate is a highly potent and selective sigma 1 (σ1) receptor ligand, displaying a Ki value of 0.08 nM for σ1 and 1377 nM for σ2. It exhibits negligible affinity for other receptors, ion channels, and enzymes.... | |||
T50090 | 3-(2-phenylethynyl)pyridine | Others | |
3-(2-phenylethynyl)pyridine is a pyridine derivative that is a ligand for a variety of receptors in the human body, including dopamine D2 receptors, sigma-1 receptors, and 5-HT6 receptors. It has been studied for the tre... | |||
T25584 | KSCM-1 | KSCM 1 | |
KSCM-1 is a selective sigma-1 receptor ligand. | |||
T26100 | RLH 033 | RLH033,RLH-033 | |
RLH 033 is a selective ligand for the sigma 1 recognition site. | |||
T16445 | PD 144418 | Sigma receptor | |
PD 144418 displays potential antipsychotic activity. PD 144418 is a high affinity, potent and selective sigma 1 (σ1) receptor ligand (Ki: 0.08 nM and 1377 nM for σ1 and σ2 respectively). It shows devoid of any significan... | |||
T61846 | CM398 | ||
CM398 is an orally active chemical compound that acts as a highly selective ligand for the sigma-2 receptor (K i =0.43 nM), demonstrating a significant ratio of selectivity between sigma-1 and sigma-2 receptors (1000-fol... |